Introduction to Industrial Drug Discovery:

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• Introduction to Industrial Drug Discovery
• From Target Finding to
• Developmental Candidates

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Goal of Drug Discovery
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• Research and Development in
• Pharmaceutical Industry

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The Research Phase
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The Development Phase
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What are Genomics/Proteomics/Bioinformatics?
How do these disciplines impact industrial drug
discovery? How can we find and validate new drug
targets?
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What ist High-Throughput Screening (HTS),
Combinatorial Chemistry, Chemoinformatics? How
can Structural Research (Xray, NMR) and
Molecular Modelling assist Lead Finding?
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Optimization Strategies in Medicinal
Chemistry What are ADMET parameters and how can
they be determined or predicted? How can
Structural Research (Xray, NMR) and Molecular
Modelling assist Lead Optimization?
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